A report on Estrogen receptor and ICI-164384

A dimer of the ligand-binding region of ERβ (PDB rendering based on ).
The domain structures of ERα and ERβ, including some of the known phosphorylation sites involved in ligand-independent regulation.
A dimer of the ligand-binding region of ERα (PDB rendering based on ).
Nolvadex (tamoxifen) 20 mg
Arimidex (anastrozole) 1 mg

It is a silent antagonist of the estrogen receptor (ER) with no intrinsic estrogenic activity and hence is a pure antiestrogen, unlike selective estrogen receptor modulators (SERMs) like tamoxifen.

- ICI-164384

Antiestrogens (e.g., fulvestrant, ICI-164384, ethamoxytriphetol)

- Estrogen receptor
A dimer of the ligand-binding region of ERβ (PDB rendering based on ).

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